Warfarin

Anticoagulants

Anticoagulants · Vitamin K antagonist

Warfarin

Dose

Start 5 mg OD (3 mg if elderly / liver disease); titrate to target INR

Mechanism

Inhibits VKORC1 → ↓ factors II, VII, IX, X and proteins C, S

Indications

  • Mechanical heart valve
  • Antiphospholipid syndrome
  • AF when DOAC contraindicated

Contraindications

  • Pregnancy (1st trimester, near delivery)
  • Active bleeding

Use

Many drug / food interactions; bridge with LMWH if rapid anticoagulation required.

Monitoring

INR — daily until stable then weekly → monthly. Target 2–3 (2.5–3.5 mechanical valve).

Side effects

  • Bleeding
  • Skin necrosis
  • Purple-toe syndrome
  • Teratogenic

Pregnancy safety

Avoid — use LMWH instead

Related in WardRound

Always confirm dose against your local formulary / BNF before prescribing.

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