Propylthiouracil

Endocrinology

Endocrinology · Thionamide (blocks T4→T3 conversion)

Propylthiouracil

Dose

200–400 mg/day divided TDS; thyroid storm 200 mg q4h PO/NG.

Use

First-trimester pregnancy hyperthyroidism and thyroid storm.

Monitoring

LFTs (hepatic failure risk), FBC, TFTs q4 wk.

Side effects

  • Hepatotoxicity
  • Agranulocytosis
  • ANCA-associated vasculitis

Related in WardRound

Always confirm dose against your local formulary / BNF before prescribing.

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