Metoprolol succinate (XL)

Cardiology

Cardiology · β₁-selective adrenergic blocker (extended release)

Metoprolol succinate (XL)

Dose

HF: 12.5–25 mg OD, double q2 weeks to 200 mg OD. Post-MI: 25–200 mg OD.

Mechanism

Selective β₁ blockade with sustained 24-h profile.

Indications

  • HFrEF
  • Post-MI secondary prevention
  • Angina
  • Rate control AF

Contraindications

  • Severe bradycardia
  • High-grade AV block
  • Acute decompensated HF
  • Cardiogenic shock

Use

Guideline β-blocker for HFrEF and post-MI.

Monitoring

HR, BP, symptoms, K+ if combined with MRA.

Side effects

  • Bradycardia
  • Hypotension
  • Fatigue
  • Depression
  • Nightmares

Pregnancy safety

Category C — labetalol preferred.

Related in WardRound

Always confirm dose against your local formulary / BNF before prescribing.

WardRound

WardRound

Clinical Decisions in Seconds