Isotretinoin

Dermatology

Dermatology · Systemic retinoid

Isotretinoin

Dose

0.5 mg/kg/day PO with food, increasing to 1 mg/kg/day; cumulative target 120–150 mg/kg.

Contraindications

  • Pregnancy
  • Concurrent tetracyclines (intracranial hypertension)

Use

Severe nodulocystic or scarring acne unresponsive to antibiotics.

Monitoring

Pregnancy test monthly, lipids and LFTs at baseline and 8 weeks, mood review.

Side effects

  • Dry lips, skin and eyes
  • Hypertriglyceridaemia
  • Myalgia
  • Mood disturbance

Pregnancy safety

Absolutely contraindicated — pregnancy prevention programme mandatory.

Always confirm dose against your local formulary / BNF before prescribing.

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